Ocaperidone
Cat. No.：YN320101
CAS No. ：129029-23-8
| 产品名称: | Ocaperidone |
| CAS No.: | 129029-23-8 |
| Chemical Name: | 3-[2-[4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-2,9-dimethyl-4H-pyrido[1,2-a]pyrimidin-4-one; R 79598 |
| Synonyms: | R79598 |
| 分子量: | 420.48 |
| 分子式: | C₂₄H₂₅FN₄O₂ |
| SMILES: | O=C1C(CCN2CCC(C3=NOC4=C3C=CC(F)=C4)CC2)=C(C)N=C5N1C=CC=C5C |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Ocaperidone 是一种有效的安定剂，为5-HT2和 多巴胺D2的拮抗剂，5-HT1A的激动剂，对 5-HT2，a1-adrenergic 受体，dopamine D2，组胺 H1和 a2-adrenergic 受体的Ki值分别为 0.14 nM，0.46 nM，0.75 nM，1.6 nM 和 5.4 nM，对 h5-HT1A的 pEC50和pKi值分别为 7.60 和 8.08。 |
| IC50和靶点: | [{name:"5-HT2 Receptor:0.14 nM (Ki)"},{name: "D2 Receptor:0.75 nM (Ki)"},{name: "5-HT1A Receptor:7.6 (pEC50, h5-HT1A)"},{name: "5-HT1A Receptor:8.08 (pKi, h5-HT1A)"},{name: "a1-adrenergic receptor:0.46 nM (Ki)"},{name: "Histamine H1:1.6 nM (Ki)"},{name: "a2-adrenergic receptor:5.4 nM (Ki)"}] |
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| Solvent & Solubility: |
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