SB-200646
Cat. No.:YN320239
产品名称: | SB-200646 |
CAS No.: | 143797-63-1 |
Chemical Name: | |
Synonyms: | SB 200646A |
分子量: | 266.30 |
分子式: | C₁₅H₁₄N₄O |
SMILES: | O=C(NC1=CC=CN=C1)NC2=CC3=C(N(C)C=C3)C=C2 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | SB-200646 是第一个对5-HT2B/2C的选择性超过 5-HT2A的拮抗剂,5-HT2B,5-HT2C和 5-HT2A的pKi值分别为 7.5、6.9 和 5.2。SB-200646 具有口服活性,在体内具有电生理和抗焦虑特性。 |
IC50和靶点: | [{name:"5-HT2B Receptor:7.5 (pKi)"},{name: "5-HT2C Receptor:6.9 (pKi)"},{name: "5-HT2A Receptor:5.2 (pKi)"}] |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |