Methiothepin mesylate
Cat. No.：YN320342
| 产品名称: | Methiothepin mesylate |
| CAS No.: | 74611-28-2 |
| Chemical Name: | |
| Synonyms: | 马来酸甲硫替平; Metitepine mesylate; Ro 8-6837 mesylate |
| 分子量: | 452.65 |
| 分子式: | C₂₁H₂₈N₂O₃S₃ |
| SMILES: | CN1CCN(C2CC3=CC=CC=C3SC4=CC=C(SC)C=C24)CC1.CS(=O)(O)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Methiothepin mesylate 是一种有效的，非选择性的5-HT2receptor拮抗剂，pKd值为 7.10 (5-HT1A)，7.28 (5HT1B)，7.56 (5HT1C)，6.99 (5HT1D)，7.0 (5-HT5A)，7.8 (5-HT5B)，8.74 (5-HT6) 和 8.99 (5-HT7)，pKi值为 8.50 (5HT2A)，8.68 (5HT2B) 和 8.35 (5HT2C)。 |
| IC50和靶点: | [{name:"5-HT1A Receptor:7.10 (pKd)"},{name: "5-HT1B Receptor:7.28 (pKd)"},{name: "5-HT1C Receptor:7.56 (pKd)"},{name: "5-HT1D Receptor:6.99 (pKd)"},{name: "5-HT5A Receptor:7.0 (pKd)"},{name: "5-HT5B Receptor:7.8 (pKd)"},{name: "5-HT6 Receptor:8.74 (pKd)"},{name: "5-HT7 Receptor:8.99 (pKd)"},{name: "5-HT2A Receptor:8.50 (pKi)"},{name: "5-HT2B Receptor:8.68 (pKi)"},{name: "5-HT2C Receptor:8.35 (pKi)"}] |
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| Clinical Trial: | |
| Solvent & Solubility: |
