Opiranserin
Cat. No.：YN320400
| 产品名称: | Opiranserin |
| CAS No.: | 1441000-45-8 |
| Chemical Name: | |
| Synonyms: | VVZ-149;VVZ-000149 |
| 分子量: | 394.51 |
| 分子式: | C₂₁H₃₄N₂O₅ |
| SMILES: | O=C(C1=CC(OC)=C(OCCCC)C(OC)=C1)NCC2(CCOCC2)N(C)C |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Opiranserin，一种非阿片类药物和非甾体抗炎止痛药，是 2 型甘氨酸转运蛋白(GlyT2)和 5-羟色胺受体2A(5HT2A)的双重拮抗剂，IC50分别为 0.86 和 1.3 μM。Opiranserin 对 rP2X3 有拮抗作用 (IC50=0.87 μM)。Opiranserin 可用于术后疼痛的研究。 |
| IC50和靶点: | [{name:"GlyT2:0.86 μM (IC50)'}, 'P2X3 Receptor', {'rP2X3:0.87 μM (IC50)"},{name: "5-HT2A Receptor:1.3 μM (IC50)"}] |
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| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
