OPC-14523 free base
Cat. No.:YN320500
产品名称: | OPC-14523 free base |
CAS No.: | 145969-30-8 |
Chemical Name: | |
Synonyms: | |
分子量: | 413.94 |
分子式: | C₂₃H₂₈ClN₃O₂ |
SMILES: | O=C1N(CCCN2CCN(C3=CC=CC(Cl)=C3)CC2)C4=C(C(OC)=CC=C4)CC1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | OPC-14523 free base 是一种具有口服活性的sigma和5-HT1A受体激动剂,对 sigma 受体 (σ1/2IC50=47/56 nM)、5-HT1A 受体 (IC50=2.3 nM) 和 5-HT 转运体 (IC50=80 nM) 具有高度亲和力。OPC-14523 free base 显示抗抑郁药样活性。 |
IC50和靶点: | [{name:"5-HT1A Receptor:2.3 nM (IC50)"},{name: "sigma 1:47 nM (IC50)"},{name: "sigma 2:56 nM (IC50)"}] |
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