Cisapride
Cat. No.：YN320823
CAS No. ：81098-60-4
| 产品名称: | Cisapride |
| CAS No.: | 81098-60-4 |
| Chemical Name: | rel-4-amino-5-chloro-N-[1-[(3R,4S)-3-(4-fluorophenoxy)propyl]-3-methoxy-4-piperidinyl]-2-methoxy-benzamide |
| Synonyms: | R 51619; (±)-Cisaprid |
| 分子量: | 465.95 |
| 分子式: | C₂₃H₂₉ClFN₃O₄ |
| SMILES: | O=C(N[C@@H]1[C@H](OC)CN(CCCOC2=CC=C(F)C=C2)CC1)C3=CC(Cl)=C(N)C=C3OC |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Cisapride(R 51619)是5-HT4受体激动剂，还是hERG抑制剂。 |
| IC50和靶点: | [{name:"5-HT4 Receptor:0.14 μM (EC50)"}] |
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| Solvent & Solubility: |
Park, J.S., Im, W., Choi, S., et al.Discovery and SAR of N-(1-((substituted piperidin-4-yl)methyl)-3-methoxypiperidin-4-yl)-2-methoxybenzamide derivatives: 5-Hydroxytryptamine receptor 4 agonist as a potent prokinetic agentEur. J. Med. Chem.109,75-88(2016)
