WAY-181187
Cat. No.:YN320855
产品名称: | WAY-181187 |
CAS No.: | 554403-49-5 |
Chemical Name: | |
Synonyms: | SAX-187 |
分子量: | 380.87 |
分子式: | C₁₅H₁₃ClN₄O₂S₂ |
SMILES: | NCCC1=CN(S(=O)(C2=C(Cl)N=C3SC=CN32)=O)C4=C1C=CC=C4 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | WAY-181187 (SAX-187) 是一种有效的选择性5-HT6受体激动剂,Ki为 2.2 nM,EC50为 6.6 nM。WAY181187 介导 5-HT6 受体依赖性信号通路,如 cAMP,Fyn 和 ERK1/2 激酶,作为特异性激动剂。 |
IC50和靶点: | [{name:"5-HT6 Receptor:2.2 nM (Ki)"},{name: "5-HT6 Receptor:6.6 nM (EC50)"}] |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |