RS-127445
Cat. No.:YN320983
产品名称: | RS-127445 |
CAS No.: | 199864-87-4 |
Chemical Name: | 4-(4-Fluoro-1-naphthalenyl)-6-(1-methylethyl)-2-pyrimidinamine; 2-Amino-4-(4-fluoronaphth-1-yl)-6-isopropylpyrimidine; MT 500; RS 127445; |
Synonyms: | MT500 |
分子量: | 281.33 |
分子式: | C₁₇H₁₆FN₃ |
SMILES: | NC1=NC(C(C)C)=CC(C2=C3C=CC=CC3=C(F)C=C2)=N1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | RS-127445 是一种有效的,具有口服活性的,高亲和力选择性5-HT2B受体拮抗剂,pKi为 9.5,比作用于其他受体和离子通道的选择性高 1000 倍。 |
IC50和靶点: | [{name:"5-HT2B Receptor:9.5 nM (pKi)"}] |
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Clinical Trial: | |
Solvent & Solubility: |