Isamoltane hemifumarate
Cat. No.：YN321231
| 产品名称: | Isamoltane hemifumarate |
| CAS No.: | 874882-92-5 |
| Chemical Name: | |
| Synonyms: | |
| 分子量: | 332.40 |
| 分子式: | C₁₆H₂₂N₂O₂.₁/₂C₄H₄O₄ |
| SMILES: | OC(COC1=CC=CC=C1N2C=CC=C2)CNC(C)C.O=C(O)/C=C/C(O)=O.[1/2] |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Isamoltane hemifumarate 是一种选择性的5-HT1B受体拮抗剂，抑制 [125I]ICYP 与大鼠脑膜中 5-HT1B识别位点结合的IC50值为 39 nM。Isamoltane hemifumarate 也是一种β-肾上腺素受体配体，IC50值为 8.4 nM。Isamoltane hemifumarate 具有抗焦虑活性。 |
| IC50和靶点: | [{name:"β-adrenoceptor:8.4 nM (IC50)"},{name: "5-HT1B Receptor:39 nM (IC50)"}] |
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