NAN-190 hydrobromide
Cat. No.:YN321247
CAS No. :115338-32-4
产品名称: | NAN-190 hydrobromide |
CAS No.: | 115338-32-4 |
Chemical Name: | 2-[4-[4-(2-methoxyphenyl)-1-piperazinyl]butyl]-1H-isoindole-1,3(2H)-dione, monohydrobromide |
Synonyms: | NAN190 hydrobromide;NAN 190 hydrobromide |
分子量: | 474.39 |
分子式: | C₂₃H₂₈BrN₃O₃ |
SMILES: | O=C1N(CCCCN2CCN(C3=CC=CC=C3OC)CC2)C(C4=C1C=CC=C4)=O.[H]Br |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | NAN-190 hydrobromide 是一种血清素受体5-HT受体拮抗剂。NAN-190 hydrobromide 是5-HT1A选择性拮抗剂。 |
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Rydelek-Fitzgerald, L., Teitler, M., Fletcher, P.W., et al.NAN-190: Agonist and antagonist interactions with brain 5-HT1A receptorsBrain Res.532(1-2),191-196(1990)
Villalobos-Molina, R., Gallardo-Ortíz, I.A., López-Guerrero, J.J., et al.Evidence that NAN-190-induced hypotension involves vascular α1-adrenoceptor antagonism in the ratEur. J. Pharmacol.455(1),59-64(2002)
Kessler, E.J., Sprouse, J., and Harrington, M.E.NAN-190 potentiates the circadian response to light and speeds re-entrainment to advanced light cyclesNeuroscience154(4),1187-1194(2008)