Alosetron (Hydrochloride(1:X))
Cat. No.：YN321294
| 产品名称: | Alosetron (Hydrochloride(1:X)) |
| CAS No.: | 132414-02-9 |
| Chemical Name: | |
| Synonyms: | GR 68755 (Hydrochloride(1:X)); GR 68755X (Hydrochloride(1:X)) |
| 分子量: | 暂无 |
| 分子式: | C₁₇H₁₈N₄O.xHCl |
| SMILES: | O=C1N(CC2=C(NC=N2)C)CCC(N3C)=C1C4=C3C=CC=C4.[F,Cl,Br,I][ClH] |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Alosetron (GR 68755) Hydrochloride(1:X) 是一种高效、高选择性的 5-HT3 受体 (5-HT3 receptor) 拮抗剂。Alosetron Hydrochloride(1:X) 用于肠易激综合征 (IBS) 的研究。Alosetron Hydrochloride(1:X) 阻断 5HT3 介导的豚鼠肌间和粘膜下神经元的快速去极化，IC50在 ~55 nM。Alosetron Hydrochloride(1:X) 减轻清醒或麻醉犬直肠扩张的内脏伤害性效应。具有抗炎 |
| IC50和靶点: | |
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| Solvent & Solubility: |
