Tianeptine
Cat. No.：YN321315
CAS No. ：72797-41-2
| 产品名称: | Tianeptine |
| CAS No.: | 72797-41-2 |
| Chemical Name: | 7-[(3-Chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoic Acid S,S-Dioxide; (+/-)-7-[(3-Chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2] |
| Synonyms: | 噻奈普汀 |
| 分子量: | 436.95 |
| 分子式: | C₂₁H₂₅ClN₂O₄S |
| SMILES: | O=C(CCCCCCNC(C1=CC=CC=C1N2C)C3=CC=C(C=C3S2(=O)=O)Cl)O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Tianeptine 是一种选择性5-HT摄取促进剂。Tianeptine 对包括 5-HT 和多巴胺 (IC50>10 μM) 在内的多种受体没有亲和力，并且对去甲肾上腺素和多巴胺的吸收没有影响。Tianeptine 具有抗抑郁，抗焦虑，镇痛和神经保护作用。 |
| IC50和靶点: | |
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| Solvent & Solubility: |
Malen, C., et al.: Experientia, 28, 811 (1972), Safa, A., et al.: J. Biol. Chem., 262, 7884 (1987), Ford, J.M., et al.: Pharmacol. Rev., 42, 155, (1990), Pierre, A., et a.: Cancer Res., 51, 2312 (1991),
