Paliperidone palmitate
Cat. No.：YN321330
| 产品名称: | Paliperidone palmitate |
| CAS No.: | 199739-10-1 |
| Chemical Name: | 9-Hydroxyrisperidone Palmitate; Invega Sustenna; RO 92670; Hexadecanoic Acid 3-[2-[4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-9-yl Ester; |
| Synonyms: | 9-Hydroxyrisperidone palmitate |
| 分子量: | 664.89 |
| 分子式: | C₃₉H₅₇FN₄O₄ |
| SMILES: | O=C(OC1CCCN(C1=NC(C)=C2CCN3CCC(C4=NOC5=C4C=CC(F)=C5)CC3)C2=O)CCCCCCCCCCCCCCC |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Paliperidone palmitate (9-Hydroxyrisperidone palmitate) 是一种非典型长效抗精神病药，是 Paliperidone 的酯类前药。Paliperidone 是一种非典型抗精神病药的多巴胺 (dopamine) 拮抗剂和5-HT2A拮抗剂。Paliperidone palmitate 对精神分裂症有效。 |
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Hough, D. et al.: Prog. Neuro-psychophamacol. Biol. Psych., 33, 1022 (2009)
Samtani, M.N. et al.: Clin. Pharmacokin., 48, 585 (2009)
Nasrallah, H.A. et al.: Neuropsychopharmacology, 35, 2072 (2010)
