Cyclobenzaprine hydrochloride
Cat. No.:YN321569
产品名称: | Cyclobenzaprine hydrochloride |
CAS No.: | 6202-23-9 |
Chemical Name: | 3-(5H-dibenzo[a,d]cyclohepten-5-ylidene)-N,N-dimethyl-1-propanamine, monohydrochloride |
Synonyms: | 盐酸环苯扎林; MK130 hydrochloride |
分子量: | 311.85 |
分子式: | C₂₀H₂₂ClN |
SMILES: | CN(C)CC/C=C1C2=CC=CC=C2C=CC3=CC=CC=C\13.Cl |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Cyclobenzaprine hydrochloride (MK130 hydrochloride) 是骨骼肌松弛剂,对中枢神经有镇静活性。 |
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Gregori-Puigjané, E., Setola, V., Hert, J., et al.Identifying mechanism-of-action targets for drugs and probesProc. Natl. Acad. Sci. USA109(28),11178-11183(2012)
Honda, M., Nishida, T., and Ono, H.Tricyclic analogs cyclobenzaprine, amitriptyline and cyproheptadine inhibit the spinal reflex transmission through 5-HT2 receptorsEur. J. Pharmacol.458(1-2),91-99(2003)
Lounkine, E., Keiser, M.J., Whitebread, S., et al.Large scale prediction and testing of drug activity on side-effect targetsNature486(7403),361-367(2012)