Pimethixene
Cat. No.：YN321609
| 产品名称: | Pimethixene |
| CAS No.: | 314-03-4 |
| Chemical Name: | |
| Synonyms: | Pimetixene |
| 分子量: | 293.43 |
| 分子式: | C₁₉H₁₉NS |
| SMILES: | CN1CC/C(CC1)=C2C3=C(SC4=C\2C=CC=C4)C=CC=C3 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Pimethixene 是抗组胺和抗血清素剂，用作抗偏头疼剂。Pimethixene 为高效的多靶点拮抗剂，对 5-HT1A，5-HT2A，5-HT2B，5-HT2C，组胺 H1，多巴胺 D2和 D4.4以及毒蕈碱 M1和 M2的pKi值分别为 7.63，10.22，10.44，8.42，10.14，8.19，7.54，8.61 和 9.38。 |
| IC50和靶点: | [{name:"5-HT2B Receptor:10.44 (pKi)"},{name: "5-HT2A Receptor:10.22 (pKi)"},{name: "5-HT2C Receptor:8.42 (pKi)"},{name: "5-HT1A Receptor:7.63 (pKi)"},{name: "M2 receptor:9.38 (pKi)"},{name: "M1 receptor:8.61 (pKi)"},{name: "D2 receptor:8.19 (pKi)"},{name: "DD4.4 receptor:7.54 (pKi)"}] |
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