Trimipramine maleate
Cat. No.：YN321629
| 产品名称: | Trimipramine maleate |
| CAS No.: | 521-78-8 |
| Chemical Name: | 10,11-dihydro-N,N,β-trimethyl-5H-dibenz[b,f]azepine-5-propanamine, (2Z)-2-butenedioate |
| Synonyms: | 三甲丙咪嗪马来酸盐 |
| 分子量: | 410.51 |
| 分子式: | C₂₄H₃₀N₂O₄ |
| SMILES: | CC(CN(C)C)CN1C2=C(C=CC=C2)CCC3=C1C=CC=C3.O=C(O)/C=C\C(O)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Trimipramine maleate 是 5-HT 受体的拮抗剂，其对 5-HT1C，5-HT2和 5-HT1A受体的 pKi值分别为 6.39，8.10，4.66。 |
| IC50和靶点: | [{name:"5-HT1C Receptor:6.39 (pKi)"},{name: "5-HT2 Receptor:8.10 (pKi)"},{name: "sPLA2:4.66 (pKi)"}] |
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Gross, G., Xin, X., and Gastpar, M.Trimipramine: Pharmacological reevaluation and comparison with clozapineNeuropharmacology30(11),1159-1166(1991)
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