L-365260
Cat. No.：YN322173
CAS No. ：118101-09-0
| 产品名称: | L-365260 |
| CAS No.: | 118101-09-0 |
| Chemical Name: | |
| Synonyms: | L 365260;L365260 |
| 分子量: | 398.46 |
| 分子式: | C24H22N4O2 |
| SMILES: | CN1C2C=CC=CC=2C(C2C=CC=CC=2)=NC(NC(NC2C=CC=C(C)C=2)=O)C1=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | L-365260 是一种口服有效的和选择性的非肽胃泌素和脑胆囊收缩素受体 (CCK-B) 拮抗剂，其Kis 值分别为 1.9 nM 和 2.0 nM。L-365260 以立体选择性和竞争性方式与豚鼠胃胃泌素和脑CCK受体相互作用。L-365260 可增强 Morphine 缓解疼痛的活性，并防止 Morphine 耐受。 |
| IC50和靶点: | |
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