Pardoprunox
Cat. No.：YN322181
| 产品名称: | Pardoprunox |
| CAS No.: | 1197334-04-5 |
| Chemical Name: | 3,5-dihydro-5-methyl-N-3-pyridinyl-benzo[1,2-b:4,5-b′]dipyrrole-1(2H)-carboxamide, monohydrochloride |
| Synonyms: | SB206553 |
| 分子量: | 328.79594 |
| 分子式: | C17H16N4O • HCl |
| SMILES: | O=C(N1C2=CC3=C(C=C2CC1)N(C)C=C3)NC4=CN=CC=C4.Cl |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | SB 206553 盐酸盐是一种高亲和力、选择性和口服活性的5-HT2B/ 5-HT2C受体拮抗剂 (对于大鼠 5-HT2B受体，pA2=8.89，对于人 5-HT2C受体，pKi=7.92)。SB 206553 具有抗焦虑活性。 |
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Kennett, G.A., Wood, M.D., Bright, F., et al.In vitro and in vivo profile of SB 206553, a potent 5-HT2C/5-HT2B receptor antagonist with anxiolytic-like propertiesBr. J. Pharmacol.117(3),427-434(1996)
