WAY208466 dihydrochloride
Cat. No.:YN322184
产品名称: | WAY208466 dihydrochloride |
CAS No.: | 1207064-61-6 |
Chemical Name: | 3-[(3-fluorophenyl)sulfonyl]-N,N-dimethyl-1H-pyrrolo[2,3-b]pyridine-1-ethanamine, dihydrochloride |
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分子量: | 420.3 |
分子式: | C17H18FN3O2S • 2HCl |
SMILES: | CN(C)CCN1C=C(S(=O)(C2=CC(F)=CC=C2)=O)C3=CC=CN=C31.Cl.Cl |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | WAY 208466 二盐酸盐是一种强效和选择性的5-HT6受体激动剂 (对于人 5-HT6受体,EC50=7.3 nM)。WAY-208466 可提高大鼠额叶皮质 GABA 水平。WAY 208466 具有抗抑郁和抗焦虑作用。 |
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Schechter, L.E., Lin, Q., Smith, D.L., et al.Neuropharmacological profile of novel and selective 5-HT6 receptor agonists: WAY-181187 and WAY-208466Neuropsychopharmacology33(6),1323-1335(2008)