NAS-181 dimesylate
Cat. No.:YN322194
CAS No. :1217474-40-2
产品名称: | NAS-181 dimesylate |
CAS No.: | 1217474-40-2 |
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分子量: | 538.63 |
分子式: | C21H34N2O10S2 |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | NAS181 是一种有效和选择性的大鼠5-HT1B受体拮抗剂,Ki值为 47 nM。NAS181 对 r5-HT1B的选择性比牛 5-HT1B受体 (Ki=630 nM) 高 13 倍。NAS181 通过抑制末端 r5-HT1B自身受体来增加 5-HT 转换和 5-HT 的突触浓度。 |
IC50和靶点: | [{name:"Rat 5-HT1B Receptor:47 nM (IC50)"}] |
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