H2L5186303
Cat. No.:YN322245
CAS No. :139262-76-3
产品名称: | H2L5186303 |
CAS No.: | 139262-76-3 |
Chemical Name: | (Z,Z)-4,4'-[1,3-phenylenebis(oxy-4,1-phenyleneimino)]bis[4-oxo-2-butenoic acid |
Synonyms: | |
分子量: | 488.5 |
分子式: | C26H20N2O8 |
SMILES: | O=C(/C=C\C(O)=O)NC(C=C1)=CC=C1OC2=CC(OC3=CC=C(NC(/C=C\C(O)=O)=O)C=C3)=CC=C2 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | H2L5186303 是一种有效且选择性的LPA2受体(溶血磷脂酸 2 受体)拮抗剂,IC50为 9 nM。 |
IC50和靶点: | [{name:"LPA2 Receptor:9 nM (IC50)"}] |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |
Fells, J.I., Tsukahara, R., Liu, J., et al.Structure-based drug design identifies novel LPA3 antagonistsBioorg. Med. Chem.17(21),7457-7464(2009)