Zolmitriptan
Cat. No.：YN322246
| 产品名称: | Zolmitriptan |
| CAS No.: | 139264-17-8 |
| Chemical Name: | 4S-[[3-[2-(dimethylamino)ethyl]-1H-indol-5-yl]methyl]-2-oxazolidinone |
| Synonyms: | BW-311C90; 311C90 |
| 分子量: | 287.4 |
| 分子式: | C16H21N3O2 |
| SMILES: | CN(C)CCC1=CNC2=CC=C(C[C@H]3COC(N3)=O)C=C21 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Zolmitriptan (BW-311C90; 311C90) 是一种5-HT1B/1D受体部分激动剂，对 5-HT1B、5-HT1D、5-HT1F 受体的Ki分别为 5.01 nM、0.63 nM 和 63.09 nM。Zolmitriptan可用于偏头痛的研究。 |
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Wurch, T., Palmier, C., Colpaert, F.C., et al.Recombinant saphenous vein 5-HT1B receptors of the rabbit: Comparative pharmacology with human 5-HT1B receptorsBr. J. Pharmacol.120(1),153-159(1997)
Gilmore, B., and Michael, M.Treatment of acute migraine headacheAm. Fam. Physician83(3),271-280(2011)
