TC LPA5 4
Cat. No.：YN322247
CAS No. ：1393814-38-4
| 产品名称: | TC LPA5 4 |
| CAS No.: | 1393814-38-4 |
| Chemical Name: | 5-(3-Chloro-4-cyclohexylphenyl)-1-(3-methoxyphenyl)-1H-pyrazole-3-carboxylic Acid; |
| Synonyms: | LPA5-IN-4; LPA5-IN4; LPA5IN4, TC-LPA5-4 |
| 分子量: | 410.89 |
| 分子式: | C23H23ClN2O3 |
| SMILES: | O=C(C1=NN(C2=CC=CC(OC)=C2)C(C3=CC=C(C4CCCCC4)C(Cl)=C3)=C1)O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | TC LPA5 4 是一种特异性非脂质LPA5(GPR92)拮抗剂。TC LPA5 4 抑制 LPA 诱导的离体人血小板 (LPA5-RH7777细胞系) 聚集，IC50为 800 nM。TC LPA5 4 对 LPA5的选择性超过 80 个其他筛选活性分子靶点。TC LPA5 4 抑制甲状腺癌细胞的增殖和迁移。 |
| IC50和靶点: | |
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| Clinical Trial: | |
| Solvent & Solubility: |
Kozian, D., et al.: Bioorg. Med. Chem. Lett., 22, 5239 (2012)
