MRS2179 tetrasodium
Cat. No.:YN322271
产品名称: | MRS2179 tetrasodium |
CAS No.: | 1454889-37-2 |
Chemical Name: | 2'-Deoxy-N6-methyladenosine 3',5'-bisphosphate tetrasodium salt; 2'-Deoxy-N-methyl-3'-adenylic Acid 5'-(Dihydrogen Phosphate) Sodium Salt (1:4); |
Synonyms: | MRS2179 tetrasodium |
分子量: | 513.16 |
分子式: | C11H13N5O9P2Na4 |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | MRS2179 tetrasodium 是一种竞争性P2Y1受体拮抗剂,对火鸡 P2Y1 受体的Kb值为 102 nM,pA2为 6.99。MRS2179 tetrasodium 对 P2Y1 的选择性高于 P2X1 (IC50=1.15 µM)、P2X3 (12.9 µM)、P2X2、P2X4、P2Y2、P2Y4 和 P2Y6 受体。MRS2179 tetrasodium 抑制血小板聚集。 |
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Boyer, J.L., et. al.: Br. J. Pharmacol., 124, 1 (1998)