SB-737050A
Cat. No.：YN322282
| 产品名称: | SB-737050A |
| CAS No.: | 149654-41-1 |
| Chemical Name: | (8R)-8-(dipropylamino)-6,7,8,9-tetrahydro-3H-benz[e]indole-2-carbonitrile, monohydrochloride |
| Synonyms: | U-92016A |
| 分子量: | 331.9 |
| 分子式: | C19H25N3 • HCl |
| SMILES: | CCCN(CCC)[C@@H](C1)CCC2=C1C(C=C(C#N)N3)=C3C=C2.Cl |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | U92016A hydrochloride 是一种代谢稳定、具有口服活性的5-HT1A受体激动剂，具有极高的内在活性。U92016A hydrochloride 以高亲和力与中国仓鼠卵巢细胞中表达的人 5-HT1A 受体结合 (Ki=0.2 nM)。 |
| IC50和靶点: | [{name:"5-HT1A Receptor:0.2 nM (Ki)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
McCall, R.B., Romero, A.G., Bienkowski, M.J., et al.Characterization of U-92016A as a selective, orally active, high intrinsic activity 5-hydroxytryptamine1A agonistJ. Pharmacol. Exp. Ther.271(2),875-883(1994)
