Tetrindole mesylate
Cat. No.:YN380353
产品名称: | Tetrindole mesylate |
CAS No.: | 170964-68-8 |
Chemical Name: | 2,3,3a,4,5,6-Hexahydro-8-cyclohexyl-1H-pyrazino[3,2,1-j,k]carbazole Mesylate; 8-Cyclohexyl-2,3,3a,4,5,6-hexahydro-1H-pyrazino[3,2,1-jk]carbazole Monomethanesulfonate |
Synonyms: | Tetrindole |
分子量: | 390.54 |
分子式: | C21H30N2O3S |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Tetrindole mesylate 是单胺氧化酶 A (MAO A) 的选择性抑制剂。Tetrindole mesylate 以竞争性方式抑制大鼠脑线粒体 MAO A,Ki值为 0.4 μM,抑制 MAO B 的 Ki为 110 μM。Tetrindole mesylate 具有抗抑郁活性。 |
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Andreeva, N. I., et al.: Eksp. Klin. Farmakol., 59, 5 (1996)
Korshunov, V. A., et al.: Eksp. Klin. Farmakol., 63, 18 (2000)