SB 218795
Cat. No.：YN322334
CAS No. ：174635-53-1
| 产品名称: | SB 218795 |
| CAS No.: | 174635-53-1 |
| Chemical Name: | (R)-[[2-Phenyl-4-quinolinyl)carbonyl]amino]-methyl Ester Benzeneacetic Acid; SB 218795 R |
| Synonyms: | |
| 分子量: | 396.44 |
| 分子式: | C25H20N2O3 |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | SB 218795 是一种有效的选择性非肽NK3受体拮抗剂，对hNK3的Ki值为 13 nM。SB 218795 对 hNK3 的选择性分别比 hNK2 和 hNK1 高 90 倍和 7000 倍。SB 218795 可以抑制NK3受体介导的兔瞳孔收缩。 |
| IC50和靶点: | [{name:"hNK3:13 nM (Ki)"},{name: "hNK2:1220 nM (Ki)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
Giardina, G.A.
et al.: Farmaco, 54, 364 (1999)
