BMS-986188
Cat. No.:YN322336
产品名称: | BMS-986188 |
CAS No.: | 1776115-10-6 |
Chemical Name: | 9-[4-[(2-bromophenyl)methoxy]phenyl]-3,4,5,6,7,9-hexahydro-3,3,6,6-tetramethyl-1H-xanthene-1,8(2H)-dione |
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分子量: | 535.5 |
分子式: | C30H31BrO4 |
SMILES: | BrC1=C(COC2=CC=C(C3C(C(CC(C)(C)C4)=O)=C4OC(CC(C)(C)C5)=C3C5=O)C=C2)C=CC=C1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | S-986188 是δ 阿片受体的选择性正变构调节剂,EC50为 0.05 μM。 |
IC50和靶点: | |
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Burford, N.T., Livingston, K.E., Canals, M., et al.Discovery, synthesis, and molecular pharmacology of selective positive allosteric modulators of the δ-opioid receptorJ. Med. Chem.58(10),4220-4229(2015)