MRS1334
Cat. No.:YN322362
产品名称: | MRS1334 |
CAS No.: | 192053-05-7 |
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分子量: | 522.55 |
分子式: | C31H26N2O6 |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | MRS1334 是一种有效的选择性人腺苷 A3(adenosine A3) 受体拮抗剂,对 hA3、rA1、rA2A的Ki分别为 2.69 nM、>100 nM、>100 nM。MRS1334 阻断 Cl-IB-MECA 的保护作用,导致明显的心动过缓和 ST 段升高。 |
IC50和靶点: | [{name:"hA3:2.69 nM (Ki)"},{name: "rA1:>100 nM (Ki)"},{name: "rA2A:>100 nM (Ki)"}] |
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