Zelatriazin
Cat. No.:YN322365
CAS No. :1929519-13-0
产品名称: | Zelatriazin |
CAS No.: | 1929519-13-0 |
Chemical Name: | 4-oxo-N-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]-1,2,3-benzotriazine-3(4H)-acetamide |
Synonyms: | TAK-041; NBI-1065846 |
分子量: | 392.3320696 |
分子式: | C18H15F3N4O3 |
SMILES: | O=C1C2=CC=CC=C2N=NN1CC(N[C@H](C3=CC=C(C=C3)OC(F)(F)F)C)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Zelatriazin (TAK-041; NBI-1065846) 是一种有效和选择性的GPR139激动剂,EC50为 22 nM。Zelatriazin 具有研究精神分裂症阴性症状的潜力。是是 |
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Reichard, H.A., Schiffer, H.H., Monenschein, H., et al.Discovery of TAK-041: A potent and selective GPR139 agonist explored for the treatment of negative symptoms associated with schizophreniaJ. Med. Chem.64(15),11527-11542(2021)