Octamylamine
Cat. No.:YN322374
产品名称: | Octamylamine |
CAS No.: | 1977-11-3 |
Chemical Name: | 6-(4-methyl-1-piperazinyl)-11H-dibenz[b,e]azepine |
Synonyms: | MP-11 |
分子量: | 291.4 |
分子式: | C19H21N3 |
SMILES: | CN(CC1)CCN1C2=NC(C=CC=C3)=C3CC4=C2C=CC=C4 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Perlapine 是一种强效的毒蕈碱型 DREADD(由被设计的活性分子特定激活的受体)激动剂。Perlapine 对hM3Dq的选择性是 hM3受体的 10000 倍以上。 |
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Seeman, P., Corbett, R., and Van Tol, H.H.Atypical neuroleptics have low affinity for dopamine D2 receptors or are selective for D4 receptorsNeuropsychopharmacology16(2),93-110(1997)
Chen, X., Choo, H., Huang, X.P., et al.The first structure-activity relationship studies for designer receptors exclusively activated by designer drugsACS Chem. Neurosci.6(3),476-484(2015)