PTAC oxalate
Cat. No.：YN322381
| 产品名称: | PTAC oxalate |
| CAS No.: | 201939-40-4 |
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| Synonyms: | |
| 分子量: | 359.46 |
| 分子式: | C14H21N3O4S2 |
| SMILES: | CCCSC1=NSN=C1[C@@H]2[C@@H]3C[N@@](CCC3)C2.OC(C(O)=O)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | PTAC oxalate 是一种选择性毒蕈碱受体 (muscarinic receptor) 配体。PTAC oxalate 是 M2 和 M4 的部分激动剂，是 M1、M3 和 M5 的拮抗剂，对于 CHO 细胞中的 hM1-5，Ki值为 0.2-2.8 nM。PTAC oxalate 减轻神经性疼痛的机械异常性疼痛并具有抗抑郁作用。 |
| IC50和靶点: | [{name:"mAChR1:0.6 nM (Ki)"},{name: "mAChR2:2.8 nM (Ki)"},{name: "mAChR3:0.2 nM (Ki)"},{name: "mAChR4:0.2 nM (Ki)"},{name: "mAChR5:0.8 nM (Ki)"}] |
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