Lumateperone
Cat. No.：YN322462
| 产品名称: | Lumateperone |
| CAS No.: | 313368-91-1 |
| Chemical Name: | 1-(4-fluorophenyl)-4-[(6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-11H-pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl]butan-1-one; ITI 007; 1-(4-Fluorophenyl)-4-[(6bR,10aS)-2,3,6b,9,10,10a-hexahydro-3-methyl-1H-pyrido[3',4':4,5]pyrrolo[1,2,3-de]qu |
| Synonyms: | ITI-007 |
| 分子量: | 393.496 |
| 分子式: | C24H28FN3O |
| SMILES: | FC1=CC=C(C(CCCN2CC[C@H]3[C@H](C4=CC=CC5=C4N3CCN5C)C2)=O)C=C1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Lumateperone (ITI-007) 是一种5-HT2A受体拮抗剂 (Ki = 0.54 nM)、突触前 D2 受体的部分激动剂和突触后 D2 受体的拮抗剂 (Ki = 32 nM)、多巴胺 D1 受体调节剂。Lumateperone 具有抗癌活性, 可用于精神分裂症等相关精神病的研究。 |
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| Solvent & Solubility: |
Corponi, F., et al.: Eur. Neuropsychopharmacol., 29, 971-985 (2019)
