Opipramol
Cat. No.:YN380381
产品名称: | Opipramol |
CAS No.: | 315-72-0 |
Chemical Name: | 4-[3-(5H-dibenz[b,f]azepin-5-yl)propyl]-1-piperazineethanol |
Synonyms: | 奥匹哌醇; Ensidon; G-33040 |
分子量: | 363.49598 |
分子式: | C23H29N3O |
SMILES: | OCCN(CC1)CCN1CCCN2C3=CC=CC=C3C=CC4=CC=CC=C42 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Opipramol (Ensidon) 是一种非典型的三环类抗抑郁试剂 (TCA)。Opipramol 主要用作 sigma (σ) 受体激动剂,可以有效地与 sigma 识别位点相互作用,Ki值为 50 nM。Opipramol 可用于广泛性焦虑症(GAD)的研究。 |
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Müller, W.E., Siebert, B., Holoubek, G., et al.Neuropharmacology of the anxiolytic drug opipramol, a sigma site ligandPharmacopsychiatry37(Suppl 3),S189-S197(2004)