PCS1055 dihydrochloride
Cat. No.：YN322489
| 产品名称: | PCS1055 dihydrochloride |
| CAS No.: | 361979-40-0 |
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| 分子量: | 485.49 |
| 分子式: | C27H34Cl2N4 |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | PCS1055 dihydrochloride 是一种有效的，选择性的竞争性毒蕈碱M4受体拮抗剂，IC50为 18.1 nM，Kd为 5.72 nM。PCS1055 dihydrochloride 抑制放射性配体 [3H]-NMS 与M4受体的结合，Ki为 6.5 nM。PCS1055 dihydrochloride 对M4受体的选择性是 M1，M3 和 M5 受体的 100 倍以上，是 M2 受体的 30 倍。PCS1055 dihydrochloride 还是一种有效的AChE抑制剂，对电鳗和人ACh |
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