MRS2365
Cat. No.:YN322513
产品名称: | MRS2365 |
CAS No.: | 436847-09-5 |
Chemical Name: | |
Synonyms: | MRS2365 |
分子量: | 483.33 |
分子式: | C13H19N5O9P2S |
SMILES: | [Na+].[Na+].[Na+].O=P([O-])([O-])OP([O-])(=O)OC[C@@]12[C@H](C2)C(N3C4C(=C(N)N=C(SC)N=4)N=C3)[C@H](O)[C@@H]1O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | MRS2365 是一种有效的选择性P2Y1受体 (EC50=0.4 nM)/[35S]GTPγS结合/β-arrestin 2募集激动剂。MRS2365 缓解了机械性异常疼痛,提高了机械灵敏度。MRS2365 对 P2Y12 或 P2Y13 受体几乎没有激动或拮抗活性。 |
IC50和靶点: | [{name:"P2Y1 Receptor:0.4 nM (EC50)"}] |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |