VCP171
Cat. No.：YN322548
| 产品名称: | VCP171 |
| CAS No.: | 53296-10-9 |
| Chemical Name: | 2-Anilinoadenosine; CV 1808; LSU 165; |
| Synonyms: | 2-Phenylaminoadenosine |
| 分子量: | 358.35216 |
| 分子式: | C16H18N6O4 |
| SMILES: | NC1=C2C(N([C@]3([H])O[C@H](CO)[C@@H](O)[C@H]3O)C=N2)=NC(NC4=CC=CC=C4)=N1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | CV1808 (2-Phenylaminoadenosine) 是一种非选择性 A2 腺苷受体 (A2 AR) 激动剂，对 A2A 和 A3 腺苷受体亚型的Ki分别为 76 和 1450 nM。 |
| IC50和靶点: | |
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Hutchison, A.J., Webb, R.L., Oei, H.H., et al.CGS 21680C, an A2 selective adenosine receptor agonist with preferential hypotensive activityJ. Pharmacol. Exp. Ther.251(1),47-55(1989)
Abiru, T., Yamaguchi, T., Watanabe, Y., et al.The antihypertensive effect of 2-alkynyladenosines and their selective affinity for adenosine A2 receptorsEur. J. Pharmacol.196(1),69-76(1991)
Choksi, N.Y., Hussain, A., and Booth, R.G.2-Phenylaminoadenosine stimulates dopamine synthesis in rat forebrain in vitro and in vivo via adenosine A2 receptorsBrain Res.761(1),151-155(1997)
Martin, G.E., Rossi, D.J., and Jarvis, M.F.Adenosine agonists reduce conditioned avoidance responding in the ratPharmacol. Biochem. Behav.45(4),951-958(1993)
