ARC 239 dihydrochloride
Cat. No.：YN322557
CAS No. ：55974-42-0
| 产品名称: | ARC 239 dihydrochloride |
| CAS No.: | 55974-42-0 |
| Chemical Name: | 2-[2-[4-(2-methoxyphenyl)-1-piperazinyl]ethyl]-4,4-dimethyl-1,3(2H,4H)-isoquinolinedione, dihydrochloride |
| Synonyms: | ARC-239;ARC239 |
| 分子量: | 480.42676 |
| 分子式: | C24H29N3O3 • 2HCl |
| SMILES: | O=C1C2=C(C(C)(C)C(N1CCN3CCN(CC3)C4=CC=CC=C4OC)=O)C=CC=C2.Cl.Cl |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | ARC 239 dihydrochloride 是一种选择性α2B/2C肾上腺素受体拮抗剂 (α2A、α2B 和 α2C 受体的pKd值分别为 5.95、7.41 和 7.56)。ARC 239 dihydrochloride 与表达人重组 a2A-、a2B- 或 a2C- 肾上腺素受体亚型的 CHO 细胞膜结合，pKi分别为 5.6、8.4 和 7.08。 |
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