Orvepitant maleate
Cat. No.:YN322563
CAS No. :579475-24-4
产品名称: | Orvepitant maleate |
CAS No.: | 579475-24-4 |
Chemical Name: | |
Synonyms: | GW823296 maleate |
分子量: | 744.7 |
分子式: | C35H39F7N4O6 |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Orvepitant maleate (GW823296 maleate) 是一种有效,选择性,口服活性且耐受性良好的neurokinin-1 (NK-1)受体拮抗剂,对人neurokinin-1受体的pKi为 10.2。Orvepitant maleate 可以穿越血脑屏障。Orvepitant maleate 可用于抑郁症和慢性顽固性咳嗽的研究。 |
IC50和靶点: | [{name:"NK1:10.2 (pKi)"}] |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |