MRS2500 tetraammonium
Cat. No.:YN322581
产品名称: | MRS2500 tetraammonium |
CAS No.: | 630103-23-0 |
Chemical Name: | (1R,2S,4S,5S)-4-[2-Iodo-6-(methylamino)-9H-purin-9-yl]-2-(phosphonooxy)-bicyclo[3.1.0]hexane-1-methanol Dihydrogen Phosphate Tetraammonium Salt |
Synonyms: | MRS2500 tetraammonium |
分子量: | 578.19 |
分子式: | C13H21IN6O8P2 |
SMILES: | N.N.N.N.CNC1=C2C(=NC(I)=N1)N(C=N2)[C@@H]3[C@@H]4[C@@]([C@@H](OP(O)(O)=O)C3)(COP(O)(O)=O)C4 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | MRS2500 tetraammonium 是一种高效、选择性和稳定的P2Y1受体拮抗剂 (Ki=0.78 nM)。MRS2500 tetraammonium 抑制 ADP 诱导的人血小板聚集,IC50值为 0.95 nM。具有抗血栓活性。 |
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Kim, H., et al.: J. Med. Chem., 46, 4974 (2003)