VU10010
Cat. No.：YN322583
CAS No. ：633283-39-3
| 产品名称: | VU10010 |
| CAS No.: | 633283-39-3 |
| Chemical Name: | |
| Synonyms: | VU10010 |
| 分子量: | 345.845 |
| 分子式: | C17H16ClN3Os |
| SMILES: | ClC1=CC=C(CNC(C2SC3=NC(=CC(C)=C3C=2N)C)=O)C=C1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | VU10010 是一种有效的，高度选择性的M4mAChR变构增强剂，EC50为 400 nM。 VU10010 与 M4mAChR的变构位点结合，增加对乙酰胆碱的亲和力，增强与 G 蛋白偶联。VU10010 会增加卡巴胆碱引起的兴奋性传导抑制，但不能抑制海马突触的传递。 |
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
