L-902688
Cat. No.：YN322584
CAS No. ：634193-54-7
| 产品名称: | L-902688 |
| CAS No.: | 634193-54-7 |
| Chemical Name: | 5-[(1E,3R)-4,4-difluoro-3-hydroxy-4-phenyl-1-buten-1-yl]-1-[6-(2H-tetrazol-5R-yl)hexyl]-2-pyrrolidinone |
| Synonyms: | |
| 分子量: | 419.5 |
| 分子式: | C21H27F2N5O2 |
| SMILES: | [H]N1C(CCCCCCN2[C@@H](/C=C/[C@](O)([H])C(F)(F)C3=CC=CC=C3)CCC2=O)=NN=N1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | L-902688 是一种有效的，选择性的，口服活性的EP4受体激动剂，Ki为 0.38 nM，EC50为 0.6 nM。L-902688 对EP4的选择性是其他EP和类前列腺素受体的 4,000 倍以上。 |
| IC50和靶点: | [{name:"EP4:0.38 nM (Ki)"},{name: "EP4:0.6 nM (EC50)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
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