6-Chloromelatonin
Cat. No.：YN322589
| 产品名称: | 6-Chloromelatonin |
| CAS No.: | 63762-74-3 |
| Chemical Name: | N-[2-(6-Chloro-5-methoxy-1H-indol-3-yl)ethyl]acetamide; 6-Chloromelatonin; |
| Synonyms: | |
| 分子量: | 266.72 |
| 分子式: | C13H15ClN2O2 |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | 6-Chloromelatonin 是一种有效的褪黑素受体 (melatonin receptor) 激动剂，具有比褪黑素更高的代谢稳定性。6-Chloromelatonin 竞争 [3H] 褪黑素 和 2-[125I]- iodomelatonin 与MT1受体的结合 (pKi分别为8.9 和 9.1)。6-Chloromelatonin 竞争 [3H] 褪黑素 与MT2受体结合 (pKi=9.77)。 |
| IC50和靶点: | [{name:"MT1:8.9 (pKi)"},{name: "MT2:9.1 (pKi)"}] |
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| Clinical Trial: | |
| Solvent & Solubility: |
