ULS 欢迎您!
ULS 欢迎您!
> 产品中心 > 抑制剂 & 激动剂 > GPCR/G Protein > 5-HT Receptor

Linoleoyl ethanolamide

Cat. No.:YN322601

  • CAS No. :68171-52-8

    • 产品资料
    • 生物活性
    • 参考文献
    • 产品名称: Linoleoyl ethanolamide
      CAS No.: 68171-52-8
      Chemical Name: N-(2-hydroxyethyl)-9Z,12Z-octadecadienamide
      Synonyms:Linoleic acid monoethanolamide
      分子量:323.5
      分子式:C20H37NO2
      SMILES:CCCCC/C=C\C/C=C\CCCCCCCC(=O)NCCO
      存储:Please store the product under the recommended conditions in theCertificate of Analysis.
      运输:Room temperature in continental US; may vary elsewhere.
      Select Batch:
      Purity: 98%
    • 产品描述: Linoleoyl ethanolamide (Linoleic acid monoethanolamide) 是一种脂肪酸乙醇酰胺。Linoleoyl ethanolamide 可弱结合CB1和CB2受体,并分别抑制[3H]CP-55,940的结合,Ki值分别为 10 和 25μM。Linoleoyl ethanolamide 在引起小鼠过氧化氢酶方面的效力是 anandamide 的4倍,并且不会延长睡眠时间。
      IC50和靶点:
      In Vitro:
      In Vivo:
      Clinical Trial:
      Solvent & Solubility:
    • Patrono, C., Rotella, C.M., Toccafondi, R.S., et al.Prostacyclin stimulates the adenylate cyclase system of human thyroid tissueProstaglandins22(1),105-115(1981)

      Schmid, P.C., Kuwae, T., Krebsbach, R.J., et al.Anandanide and other N-acylethanolamines in mouse peritoneal macrophagesChem. Phys. Lipids87,103-110(1997)

      Lin, S., Khanolkar, A.D., Fan, P., et al.Novel analogues of arachidonylethanolamide (anandamide): Affinities for the CB1 and CB2 cannabinoid receptors and metabolic stabilityJ. Med. Chem.41(27),5353-5361(1998)

      Watanabe, K., Matsunaga, T., Nakamura, S., et al.Pharmacological effects in mice of anandamide and its related fatty acid ethanolamides, and enhancement of cataleptogenic effect of anandamide by phenylmethylsulfonyl fluorideBiol. Pharm. Bull.22(4),366-370(1999)

      Berdyshev, E.V., Schmid, P.C., Krebsbach, R.J., et al.Cannabinoid-receptor-independent cell signalling by N-acylethanolaminesBiochem. J.360,67-75(2001)

      Maccarrone, M., van der Stelt, M., Rossi, A., et al.Anandamide hydrolysis by human cells in culture and brainJ. Biol. Chem.273,32332-32339(1998)

      Bisogno, T., Maurelli, S., Melck, D., et al.Biosynthesis, uptake, and degradation of anandamide and palmitoylethanolamide in leukocytesJ. Biol. Chem.272,3315-3323(1997)

    • 摩尔计算器
    • 稀释计算器
    摩尔浓度计算器方程 :
    Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

    计算

    质量 浓度 体积 分子量
    稀释计算器 :
    Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)
    • C1
      V1
      C2
      V2
    • 您最近查看的产品:
    相关产品


    ULS 的所有产品和服务仅用于科学研究,我们不为任何其他用途提供产品和服务(也不为任何个人提供产品和服务)Copyright © 2020-2021 ULS. All Rights Reserved. 备案号:粤ICP备2021013238号-1
    0.344813s