Butaprost
Cat. No.：YN322611
CAS No. ：69685-22-9
| 产品名称: | Butaprost |
| CAS No.: | 69685-22-9 |
| Chemical Name: | 9-oxo-11α,16S-dihydroxy-17-cyclobutyl-prost-13E-en-1-oic acid, methyl ester |
| Synonyms: | |
| 分子量: | 408.6 |
| 分子式: | C24H40O5 |
| SMILES: | O=C1[C@H](CCCCCCC(OC)=O)[C@@H](/C=C/C[C@H](O)C2(CCC2)CCC)C(O)C1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Butaprost 是一种选择性前列腺素 E 受体 (EP2) 激动剂，对鼠类EP2受体的EC50值为 33 nM，Ki值为 2.4 μM。Butaprost 对鼠类 EP1，EP3 和 EP4 受体的活性较低。Butaprost 通过阻碍TGF-β/Smad2信号传导来减轻纤维化。 |
| IC50和靶点: | |
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| Clinical Trial: | |
| Solvent & Solubility: |
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