Metoclopramide hydrochloride
Cat. No.:YN322621
产品名称: | Metoclopramide hydrochloride |
CAS No.: | 7232-21-5 |
Chemical Name: | 4-amino-5-chloro-N-[2-(diethylamino)ethyl]-2-methoxy-benzamide, monohydrochloride |
Synonyms: | 盐酸甲氧氯普胺 |
分子量: | 336.3 |
分子式: | C14H22ClN3O2 • HCl |
SMILES: | ClC1=CC(C(NCCN(CC)CC)=O)=C(OC)C=C1N.Cl |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Metoclopramide hydrochloride 是一种有效和具有口服活性的5-HT3和多巴胺D2受体拮抗剂,IC50值分别为 308 nM 和 483 nM。Metoclopramide hydrochloride 可用于恶心呕吐、胃食管反流和胃轻瘫的研究。 |
IC50和靶点: | [{name:"5-HT3 Receptor:308 nM (IC50)"},{name: "D2 Receptor:483 nM (IC50)"}] |
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