(R)-Carvedilol-d
Cat. No.：YN322643
| 产品名称: | (R)-Carvedilol-d |
| CAS No.: | 80259-18-3 |
| Chemical Name: | |
| Synonyms: | MMV006172 |
| 分子量: | 368.48 |
| 分子式: | C24H24N4 |
| SMILES: | CN1CCN(CC1)C2=CC=C(NC3=C4C=CC=CC4=NC5=CC=CC=C35)C=C2 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | JP1302 是一种选择性的、高亲和力的 α2C肾上腺受体 (α2C-adrenoceptor) 的拮抗剂，其对人类 α2C受体的Kb值为 16 nM，Ki为 28 nM。JP1302 具有抗抑郁和类抗精神病作用。JP1302 可用于神经精神障碍和肾功能障碍的研究。 |
| IC50和靶点: | [{name:"human α2C-adrenoceptor:28±2 nM (Ki)"},{name: "human α2B-adrenoceptor:1470±130 nM (Ki)"},{name: "human α2A-adrenoceptor:3150±50 nM (Ki)"},{name: "rodent α2D-adrenoceptor:1700±200 nM (Ki)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
