AMN082 free base
Cat. No.：YN322652
CAS No. ：83027-13-8
| 产品名称: | AMN082 free base |
| CAS No.: | 83027-13-8 |
| Chemical Name: | |
| Synonyms: | AMN082;AMN-082 |
| 分子量: | 392.54 |
| 分子式: | C28H28N2 |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | AMN082 free base 是一种选择性，具有口服活性，可透过血脑屏障的mGluR7激动剂，通过跨膜区的变构位点直接激活受体信号。在表达mGluR7的转染哺乳动物细胞上，AMN082 free base 有效抑制 cAMP 积累并刺激 GTPγS 结合 (EC50, 64-290 nM)。AMN082 free base 对其他mGluR亚型和选择性离子型谷氨酸受体具有选择性。具有抗抑郁作用。 |
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
