Didesmethyl cariprazine
Cat. No.:YN322657
产品名称: | Didesmethyl cariprazine |
CAS No.: | 839712-25-3 |
Chemical Name: | N-[trans-4-[2-[4-(2,3-Dichlorophenyl)-1-piperazinyl]ethyl]cyclohexyl]urea |
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分子量: | 399.36 |
分子式: | C19H28Cl2N4O |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Didesmethyl cariprazine 是 Cariprazine 的代谢物,作为主要的循环活性部分。Didesmethyl cariprazine 的半衰期较长,为 1-3 周。Cariprazine是一种新型抗精神病候选活性分子,能结合 D3, D2和 5-HT1A。 |
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Gruender, G.: Curr. Opin. Invest. Drugs, 11, 823 (2010)
Seneca, N. et al.: Psychopharmacology, 218, 579 (2011)
Kiss, B. et al.: J. Pharmacol. Exp. Therap., 333, 328 (2010)