GSK256073
Cat. No.:YN322666
CAS No. :862892-90-8
产品名称: | GSK256073 |
CAS No.: | 862892-90-8 |
Chemical Name: | |
Synonyms: | GSK256073 |
分子量: | 256.69 |
分子式: | C10H13ClN4O2 |
SMILES: | O=C(N(C1=C2NC(Cl)=N1)CCCCC)NC2=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | GSK256073 是一种有效的、选择性的、口服活性的GPR109A激动剂,是一种持久的HCA2激动剂,其pEC50为 7.5 (Human HCA2)。GSK256073 可通过抑制脂降解而明显改善葡萄糖稳态,具有研究 2 型糖尿病 (T2DM) 和血脂异常的潜力。 |
IC50和靶点: | |
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Clinical Trial: | |
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